Forschung & Innovation
Publikationen
Discovery of Potent Soluble Epoxide Hydrolase (sEH) Inhibitors by Pharmacophore-Based Virtual Screening.
PMU Autor*innen
Veronika Temml, Daniela Brigitte Schuster
Alle Autor*innen
Birgit Waltenberger, Ulrike Garscha, Veronika Temml, Josephine Liers, Oliver Werz, Daniela Brigitte Schuster, Hermann Stuppner
Fachzeitschrift
JOURNAL OF CHEMICAL INFORMATION AND MODELING
Kurzfassung
Keywords
IN-VITRO, PROTEIN DATA-BANK, HIGHLY POTENT, IMPROVED PHARMACOKINETIC PROPERTIES, EPOXYGENASE-DERIVED EICOSANOIDS, UREA-BASED INHIBITORS, EPOXYEICOSATRIENOIC ACIDS, 1,3-DISUBSTITUTED UREAS, INFLAMMATORY PAIN, WATER SOLUBILITY