Paracelsus Medizinische Privatuniversität (PMU)

Forschung & Innovation
Publikationen

Heterodimeric GW7604 Derivatives: Modification of the Pharmacological Profile by Additional Interactions at the Coactivator Binding Site.

#2021
#JOURNAL OF MEDICINAL CHEMISTRY

PMU Autor*in
Daniela Brigitte Schuster

Alle Autor*innen
Alexandra K Knox, Christina Kalchschmid, Daniela Brigitte Schuster, Francesca Gaggia, Ronald Gust

Fachzeitschrift
JOURNAL OF MEDICINAL CHEMISTRY

Kurzfassung

Keywords

DETERMINANTS, BREAST-CANCER, STRUCTURAL BASIS, ACID, ESTROGEN-RECEPTOR-ALPHA, DEGRADER SERD, ANTIESTROGENS, TAMOXIFEN, MODE, MODULATORS