Research & Innovation
Publications
Heterodimeric GW7604 Derivatives: Modification of the Pharmacological Profile by Additional Interactions at the Coactivator Binding Site.
PMU Author
Daniela Brigitte Schuster
All Authors
Alexandra K Knox, Christina Kalchschmid, Daniela Brigitte Schuster, Francesca Gaggia, Ronald Gust
Journal association
JOURNAL OF MEDICINAL CHEMISTRY
Abstract
Keywords
DETERMINANTS, BREAST-CANCER, STRUCTURAL BASIS, ACID, ESTROGEN-RECEPTOR-ALPHA, DEGRADER SERD, ANTIESTROGENS, TAMOXIFEN, MODE, MODULATORS