Paracelsus Medizinische Privatuniversität (PMU)

Research & Innovation
Publications

Heterodimeric GW7604 Derivatives: Modification of the Pharmacological Profile by Additional Interactions at the Coactivator Binding Site.

#2021
#JOURNAL OF MEDICINAL CHEMISTRY

PMU Author
Daniela Brigitte Schuster

All Authors
Alexandra K Knox, Christina Kalchschmid, Daniela Brigitte Schuster, Francesca Gaggia, Ronald Gust

Journal association
JOURNAL OF MEDICINAL CHEMISTRY

Abstract

Keywords

DETERMINANTS, BREAST-CANCER, STRUCTURAL BASIS, ACID, ESTROGEN-RECEPTOR-ALPHA, DEGRADER SERD, ANTIESTROGENS, TAMOXIFEN, MODE, MODULATORS