Paracelsus Medizinische Privatuniversität (PMU)

Research & Innovation
Publications

Discovery of a benzenesulfonamide-based dual inhibitor of microsomal prostaglandin E

#2018
#EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

PMU Authors
Veronika Temml, Daniela Brigitte Schuster

All Authors
Sun-Yee Cheung, Markus Werner, Lucia Esposito, Fabiana Troisi, Vincenza Cantone, Stefanie Liening, Stefanie König, Jana Gerstmeier, Andreas Koeberle, Rossella Bilancia, Roberta Rizza, Antonietta Rossi, Fiorentina Roviezzo, Veronika Temml, Daniela Brigitte Schuster, Hermann Stuppner, Manfred Schubert-Zsilavecz, Oliver Werz, Thomas Hanke, Simona Pace

Journal association
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Abstract

Keywords

PROTEIN, IN-VIVO, VALIDATION, EFFICIENCY, OPTIMIZATION, LEUKOTRIENE BIOSYNTHESIS, MPGES-1, ANTIINFLAMMATORY DRUGS, PIRINIXIC ACID-DERIVATIVES, ARRIVE GUIDELINES